Acute Porphyria Drugs

Monograph

C01CA01 - Etilefrine
Propably not porphyrinogenic
PNP

Rationale
Non-CYP metabolism. No data pointing to CYP-interaction.
Chemical description
Structurally related to endogenous adrenaline, lacking one catechol-hydroxy moiety, and N-ethyl substituent instead of N-methy.
Therapeutic characteristics
Adrenergic substance used in hypotension.
Metabolism and pharmacokinetics
Metabolized by conjugation to sulfates and glucuronides and by deamination to hydroxymandelic acid.
Personal communication
None
Published experience
None
Similar drugs
Explore alternative drugs in similar therapeutic classes C01C / C01CA or go back.
References
Tradenames

Effortil Efortil Effortil Effortil · Etilefrine · Thomasin Effortil Effortil Effortil Effortil Effortil
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